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Pelanserin (TR2515) is a chemical compound that acts as an
antagonist
An antagonist is a character in a story who is presented as the main enemy or rival of the protagonist and is often depicted as a villain.5-HT2 and α1-adrenergic receptors.
Pelanserin (3) can be synthesized by a reaction between
Synthesis
Pelanserin (3) can be synthesized by a reaction between isatoic anhydride
Isatoic anhydride is an organic compound derived from anthranilic acid. A white solid, it is prepared by reaction of anthranilic acid with phosgene.
Reactions
Hydrolysis gives carbon dioxide and anthranilic acid. Alcoholysis proceeds similarly, ...
(1) and 1-(3-aminopropyl)-4-phenylpiperazine (2) in the presence of phosgene
Phosgene is an organic chemical compound with the formula . It is a toxic, colorless gas; in low concentrations, its musty odor resembles that of freshly cut hay or grass. It can be thought of chemically as the double acyl chloride analog of ...
.Horacio Vidrio, (1975 to Bayer Corp).
See also
*Ketanserin
Ketanserin, sold under the brand name Sufrexal, is an antihypertensive agent which is used to treat arterial hypertension and vasospasm, vasospastic disorders. It is also used in scientific research as an antiserotonergic medication, agent in th ...
References
5-HT2 antagonists Alpha-1 blockers {{pharma-stub