Phenylbutynamine (4-phenylbut-3-yn-2-amine; development code PAL-874) is a
monoamine releasing agent
A monoamine releasing agent (MRA), or simply monoamine releaser, is a drug that induces the release of one or more monoamine neurotransmitters from the presynaptic neuron into the synapse, leading to an increase in the extracellular concentrati ...
(MRA) of the
arylalkylamine family related to
β-phenethylamine
Phenethylamine (PEA) is an organic compound, natural monoamine alkaloid, and trace amine, which acts as a central nervous system stimulant in humans. In the brain, phenethylamine regulates monoamine neurotransmission by binding to trace ami ...
and
amphetamine
Amphetamine (contracted from Alpha and beta carbon, alpha-methylphenethylamine, methylphenethylamine) is a central nervous system (CNS) stimulant that is used in the treatment of attention deficit hyperactivity disorder (ADHD), narcolepsy, an ...
.
It acts as a
norepinephrine–dopamine releasing agent
A norepinephrine–dopamine releasing agent (NDRA) is a type of drug which induces the synapse, release of norepinephrine (and epinephrine) and dopamine in the body and/or brain. Many of these are amphetamine type stimulants.
Examples
Examples ...
(NDRA), albeit with far lower
potency
Potency may refer to:
* Potency (pharmacology), a measure of the activity of a drug in a biological system
* Virility
* Cell potency, a measure of the differentiation potential of stem cells
* In homeopathic dilutions, potency is a measure of ho ...
than β-phenethylamine or amphetamine.
See also
*
Phenylbutenamine
*
Phenylpropylamine
References
External links
4-Phenylbut-3-yn-2-amine (PAL-874)
Arylalkylamines
Norepinephrine-dopamine releasing agents
Partial monoamine releasing agents
Phenyl compounds
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