Nipecotic acid is a
GABA
GABA (gamma-aminobutyric acid, γ-aminobutyric acid) is the chief inhibitory neurotransmitter in the developmentally mature mammalian central nervous system. Its principal role is reducing neuronal excitability throughout the nervous system.
GA ...
uptake inhibitor used in scientific research.
Nipecotic acid has very little to no BBB penetration itself but structural modifications can be done to improve this.
See also
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Deramciclane
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Tiagabine
Tiagabine, sold under the brand name Gabitril, is an anticonvulsant medication produced by Cephalon that is used in the treatment of epilepsy. The drug is also used off-label in the treatment of anxiety disorders including panic disorder.
Medi ...
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Niacin
Nicotinic acid, or niacin, is an organic compound and a vitamer of vitamin B3, an essential human nutrient. It is produced by plants and animals from the amino acid tryptophan.
Nicotinic acid is also a prescription medication. Amounts f ...
References
3-Piperidinyl compounds
GABA reuptake inhibitors
Glycine receptor antagonists
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