MRS7292 is an experimental drug which acts as both a selective agonist of the
adenosine A3 receptor with moderate affinity, and also a
dopamine reuptake inhibitor
A dopamine reuptake inhibitor (DRI) is a class of drug which acts as a reuptake inhibitor of the monoamine neurotransmitter dopamine by blocking the action of the dopamine transporter (DAT). Reuptake inhibition is achieved when extracellular dop ...
, showing that these disparate mechanisms of action can both be produced in the same molecule.
See also
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MRS8209
MRS8209 is an experimental drug which acts as a potent, peripherally selective 5-HT2B receptor antagonist with high selectivity over other serotonin receptor
5-HT receptors, 5-hydroxytryptamine receptors, or serotonin receptors, are a group ...
References
Experimental drugs
Thiophenes
Purines
Diols
Methyl esters
Secondary amines
Chloroarenes
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