KML-010 is a
drug derived from
spiperone
Spiperone (Spiroperidol; brand name: Spiropitan ( JP)) is a typical antipsychotic and research chemical belonging to the butyrophenone chemical class. It is licensed for clinical use in Japan as a treatment for schizophrenia. Additionally, spip ...
. It functions as a highly selective
5-HT2A receptor antagonist, with negligible affinity for the
5-HT1A or
5-HT2C receptors, and over 400-fold lower affinity for the
D2 receptor in comparison to
spiperone
Spiperone (Spiroperidol; brand name: Spiropitan ( JP)) is a typical antipsychotic and research chemical belonging to the butyrophenone chemical class. It is licensed for clinical use in Japan as a treatment for schizophrenia. Additionally, spip ...
.
See also
*
Spiperone
Spiperone (Spiroperidol; brand name: Spiropitan ( JP)) is a typical antipsychotic and research chemical belonging to the butyrophenone chemical class. It is licensed for clinical use in Japan as a treatment for schizophrenia. Additionally, spip ...
References
5-HT2A antagonists
Fluoroarenes
Aromatic ketones
Spiro compounds
Imidazolidinones
{{nervous-system-drug-stub